An Improved, Scalable Synthesis of the Selective Serotonin 2A Receptor Agonist 25CN-NBOH

نویسندگان

چکیده

Abstract 4-{2-[(2-hydroxybenzyl)amino]ethyl}-2,5-dimethoxybenzo­nitrile (25CN-NBOH) was first reported as a potent and highly selective serotonin 2A receptor (5-HT2AR) agonist in 2014. The compound has since found extensive use pharmacological tool variety of vivo vitro studies. In the present study, we an improved scalable synthesis 25CN-NBOH making this readily available to scientific community.

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ژورنال

عنوان ژورنال: SynOpen

سال: 2021

ISSN: ['2509-9396']

DOI: https://doi.org/10.1055/a-1524-4439